沸点 :
497.7° C at 760 mmHg (Predicted)
密度 :
~1.2 g/cm3 (Predicted)
折射率 :
n20D 1.61 (Predicted)
IC50 :
SR-1B: IC50 = 0.50 nM (human); SR-1D: IC50 = 2.95 nM (human); SR-2C: IC50 = 7.3 nM (human); SR-3A: IC50 = 9.3 nM (human); SR-5A: IC50 = 501.19 nM (human)
Ki 数据 :
SR-1B: Ki= 5.5 nM (human); SR-2a: Ki= 7.3 nM (human); D2DR: Ki>218 nM (human); SR-1A: Ki= 230 nM (human); SR-1D: Ki= 376 nM (human)
pK值 :
pKa: 11.31 (Predicted), pKb: 9.49 (Predicted)