Date published: 2025-9-8

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PIK-III (CAS 1383716-40-2)

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说明书
CAS号码:
1383716-40-2
分子量:
319.36
分子式:
C17H17N7
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.

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PIK-III (CAS 1383716-40-2) 参考文献

  1. 选择性 VPS34 抑制剂可阻止自噬,并揭示 NCOA4 在体内铁蛋白降解和铁稳态中的作用。  |  Dowdle, WE., et al. 2014. Nat Cell Biol. 16: 1069-79. PMID: 25327288
  2. 消除VPS34抑制。  |  Marsh, T. and Debnath, J. 2015. Nat Cell Biol. 17: 1-3. PMID: 25679028
  3. 抑制人类I类与III类磷脂酰肌醇3'-激酶。  |  Hassett, MR., et al. 2017. Biochemistry. 56: 4326-4334. PMID: 28719179
  4. 2,5-己二酮通过PI3K/Akt/mTOR途径诱导VSC4.1细胞自噬死亡。  |  Guan, H., et al. 2017. Mol Biosyst. 13: 1993-2005. PMID: 28752163
  5. 用小分子靶向禁止素促进黑色素瘤细胞的黑色素生成和凋亡。  |  Djehal, A., et al. 2018. Eur J Med Chem. 155: 880-888. PMID: 29960207
  6. 使用第二代自噬抑制剂靶向静止期白血病干细胞。  |  Baquero, P., et al. 2019. Leukemia. 33: 981-994. PMID: 30185934
  7. 巨噬细胞向吞噬体金黄色葡萄球菌输送营养物质,支持细菌生长。  |  Flannagan, RS. and Heinrichs, DE. 2020. EMBO Rep. 21: e50348. PMID: 32452129
  8. RKO 癌细胞对 VPS34 依赖性的基础是铁依赖性代谢脆弱性。  |  Kobylarz, MJ., et al. 2020. PLoS One. 15: e0235551. PMID: 32833964
  9. MLN4924抑制刺猬信号通路并激活自噬以减轻小鼠激光诱导的脉络膜新生血管病变。  |  Xie, L., et al. 2020. Biomed Pharmacother. 130: 110654. PMID: 34321162
  10. 将自噬作为治疗小儿急性淋巴细胞白血病的策略。  |  Bwanika, HC., et al. 2024. Sci Rep. 14: 4000. PMID: 38369625

订购信息

产品名称产品编号规格价格数量收藏夹

PIK-III, 5 mg

sc-507530
5 mg
RMB1918.00