IC50 :
Trypanosoma brucei rhodesiense: IC50 = 5.37 µM; Trypanosoma brucei: IC50 = 5.4 µM; Plasmodium falciparum: IC50 >200 µM; Entamoeba histolytica: IC50 = 200 µM; Leishmania donovani: IC50 >200 µM
Ki 数据 :
Hypoxanthine-guanine phosphoribosyltransferase: Ki= 126 µM (Trypanosoma brucei brucei)
pK值 :
pKa: 1.46 (Predicted), pKb: 9.42 (Predicted)