Date published: 2025-9-6

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A-443654 (CAS 552325-16-3)

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备用名:
αS-[[[5-(3-methyl-1H-indazol-5-yl)-3-pyridinyl]oxy]methyl]-1H-indole-3-ethanamine, (2S)-1-(1H-indol-3-yl)-3-[5-(3-methyl-2H-indazol-5-yl)pyridin-3-yl]oxypropan-2-amine
CAS号码:
552325-16-3
分子量:
397.5
分子式:
C24H23N5O
For Research Use Only. Not Intended for Diagnostic or Therapeutic Use.

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A-443654 (CAS 552325-16-3) 参考文献

  1. 抑制 Akt 可抑制胶质母细胞瘤和胶质母细胞瘤干样细胞的生长。  |  Gallia, GL., et al. 2009. Mol Cancer Ther. 8: 386-93. PMID: 19208828
  2. 抑制剂劫持 Akt 激活。  |  Okuzumi, T., et al. 2009. Nat Chem Biol. 5: 484-93. PMID: 19465931
  3. Akt 抑制剂可诱导慢性淋巴细胞白血病细胞凋亡。  |  de Frias, M., et al. 2009. Haematologica. 94: 1698-707. PMID: 19815839
  4. Akt 抑制剂与拓扑异构酶毒药之间的拮抗作用与环境有关。  |  Gálvez-Peralta, M., et al. 2014. Mol Pharmacol. 85: 723-34. PMID: 24569089
  5. TORC2:治疗老年性记忆障碍的新靶点。  |  Johnson, JL., et al. 2015. Sci Rep. 5: 15193. PMID: 26489398
  6. 极光激酶 A 促进乙型肝炎病毒的复制和表达。  |  Jeong, GU. and Ahn, BY. 2019. Antiviral Res. 170: 104572. PMID: 31376425
  7. 基于张量分解无监督特征提取的新型冠状病毒(SARS-CoV-2)先进硅学药物发现新方法。  |  Taguchi, YH. and Turki, T. 2020. PLoS One. 15: e0238907. PMID: 32915876
  8. AKT调节剂A-443654可减少α-突触核蛋白的表达,并使ER应激和自噬正常化。  |  Gandelman, M., et al. 2021. J Biol Chem. 297: 101191. PMID: 34520759
  9. 机器学习筛选出针对与肝细胞癌增殖相关的预后基因信号的潜在药物  |  Liu, J., et al. 2022. Front Genet. 13: 900380. PMID: 35836576
  10. 玉竹酮通过上调 AKT/GSK-3β/β-catenin 信号刺激斑马鱼幼体的骨矿化,并促进间充质干细胞的成骨分化。  |  Zhong, YT., et al. 2023. J Orthop Translat. 40: 132-146. PMID: 37457309

订购信息

产品名称产品编号规格价格数量收藏夹

A-443654, 1 mg

sc-507339
1 mg
RMB1579.00