Peg10 Inhibitors refer to a diverse class of chemical compounds designed to target and modulate the activity of the PEG10 gene, primarily by interfering with its expression or function. PEG10, which stands for Paternally Expressed Gene 10, is a unique imprinted gene in mammals, implicated in various cellular processes, including cell proliferation, apoptosis, and cancer development. Inhibitors within this class act as valuable tools for researchers and scientists to investigate the intricate mechanisms through which PEG10 influences these processes. These compounds exhibit diverse chemical structures and mechanisms of action, enabling a comprehensive exploration of PEG10's roles in cellular biology.
The mechanisms by which Peg10 Inhibitors function can vary widely. Some compounds focus on epigenetic regulation, impacting PEG10 gene expression by targeting DNA methylation or histone modifications within its regulatory regions. Others may affect post-transcriptional processing, mRNA stability, or translation of PEG10 transcripts. Additionally, Peg10 Inhibitors can potentially interfere with the interactions between PEG10 and its downstream targets, inhibiting specific cellular pathways or signaling cascades associated with PEG10 function. By providing a suite of chemical tools to manipulate PEG10, this class of inhibitors empowers researchers to unravel the complex web of molecular events associated with PEG10's role in normal cellular physiology and disease states. Understanding the mechanisms and consequences of PEG10 inhibition can pave the way for new insights into the fundamental biology of this gene and its potential implications in various biological contexts.
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| Nombre del producto | NÚMERO DE CAS # | Número de catálogo | Cantidad | Precio | MENCIONES | Clasificación |
|---|---|---|---|---|---|---|
Zebularine | 3690-10-6 | sc-203315 sc-203315A sc-203315B | 10 mg 25 mg 100 mg | ¥1422.00 ¥3136.00 ¥11101.00 | 3 | |
La zebularina es un inhibidor de la ADN metiltransferasa que impide la metilación de la región promotora de PEG10, lo que conduce a una reducción de la expresión del gen PEG10. | ||||||
5-Aza-2′-Deoxycytidine | 2353-33-5 | sc-202424 sc-202424A sc-202424B | 25 mg 100 mg 250 mg | ¥2414.00 ¥3565.00 ¥4716.00 | 7 | |
Este inhibidor, también conocido como Decitabina, actúa de forma similar a la Zebularina inhibiendo las ADN metiltransferasas y desmetilando el promotor de la PEG10. | ||||||
RG 108 | 48208-26-0 | sc-204235 sc-204235A | 10 mg 50 mg | ¥1444.00 ¥5697.00 | 2 | |
RG108 es una pequeña molécula inhibidora de las metiltransferasas del ADN, incluidas las implicadas en la metilación del promotor de PEG10. | ||||||
Scriptaid | 287383-59-9 | sc-202807 sc-202807A | 1 mg 5 mg | ¥711.00 ¥2019.00 | 11 | |
Scriptaid es un inhibidor de la histona deacetilasa (HDAC) que modula la regulación epigenética, afectando indirectamente a la expresión de PEG10. | ||||||
5-Azacytidine | 320-67-2 | sc-221003 | 500 mg | ¥3159.00 | 4 | |
Este análogo de la citidina se incorpora al ADN e inhibe las metiltransferasas del ADN, afectando a la metilación del promotor de PEG10. | ||||||
Valproic Acid | 99-66-1 | sc-213144 | 10 g | ¥959.00 | 9 | |
El ácido valproico es un inhibidor de HDAC que puede influir en la expresión de PEG10 alterando los patrones de acetilación de las histonas. | ||||||
UNC0638 | 1255580-76-7 | sc-397012 | 10 mg | ¥3554.00 | ||
UNC0638 es un inhibidor de la histona metiltransferasa G9a, que influye indirectamente en la expresión de PEG10 a través de cambios en la metilación de las histonas. | ||||||
EPZ6438 | 1403254-99-8 | sc-507456 | 1 mg | ¥745.00 | ||
EPZ-6438 es un inhibidor de la histona metiltransferasa EZH2 que modula la expresión de PEG10 al afectar a los patrones de metilación de las histonas. | ||||||